氯法齐明

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氯法齐明

商 品 名:氯法齐明
通 用 名:
公司名称:

药物分类:抗麻风病药
药品名:氯法齐明Clofazimine

别名:氯苯吩嗪,LAMPRENE,B663

作用与用途:对麻风杆菌和其他的一些分支杆菌有抑菌作用。口服吸收不完全,吸收程度与药物粒度和剂型密切有关。吸收后,迅速进入各组织,在血流中浓度甚低,自组织中释放很慢,其消除半衰期约为70天。有约1%的药物由尿排出,有少量药物自汗腺、乳腺和皮脂腺排出。对于瘤型麻风和其他型麻风均有一定疗效,对耐砜类药物麻风杆菌感染也有效。虽然尚未发现对本品的耐药菌,但在一般情况下,应与氨苯砜联合应用。还可与利福平或乙硫异烟胺联合应用以制服耐砜类药物的菌。还对麻风反应有一定疗效,可用于因用其他药物而引起急性麻风反应的病例。此外,尚对慢性盘状红斑狼疮、掌庶脓疱角化病、皮肤溃疡,坏疽性脓皮病也有一定疗效。